GW0742 is a synthetic drug that switches on PPAR-delta, a receptor involved in how the body handles fat. GlaxoSmithKline made it in the same research program as cardarine (GW501516); it has been studied in cells and animals, and it is not approved for people.
Also known as: GW610742, GW-0742.
For GW0742, there is no approved product and no published human trial, so there are no label strengths or studied human amounts.
GW0742 is not approved anywhere we could find, and we found no product in FDA's Drugs@FDA database. GSK chemists described it in 2003, alongside GW501516, as a selective PPAR-delta activator (Sznaidman 2003).
WADA bans PPAR-delta agonists as a class under "metabolic modulators" (S4.4.1), in and out of competition; its 2026 list names GW1516 (cardarine) as an example. For what is known about the risks of this drug class, see the cardarine page.
We found no published human trial of GW0742 that we could cite.
We could not find a published human half-life or time to peak, so we do not list one. Figures quoted online usually come from animal studies or computer models.
How Dose Track handles peptides · Reconstitution calculator · Half-life calculator